Appendix B: Antiretroviral Drugs Available in Canada
Part of A Practical Guide to HIV Drug Treatment for People Living With HIV
From Canadian AIDS Treatment Information Exchange
2011
| Fusion Inhibitor |
| Common Name |
Brand Name |
Manufacturer |
| T-20, enfuvirtide |
Fuzeon |
Roche |
| Co-Receptor Inhibitor |
| Common Name |
Brand Name |
Manufacturer |
| maraviroc |
Celsentri |
ViiV Healthcare (formerly Pfizer) |
| Nukes (Nucleoside and Nucleotide Analogues, or NRTIs) |
| Common Name |
Brand Name |
Manufacturer |
| abacavir, ABC |
Ziagen |
ViiV Healthcare (formerly GlaxoSmithKline) |
| AZT, zidovudine |
Retrovir |
ViiV Healthcare (formerly GlaxoSmithKline) |
| d4T, stavudine |
Zerit |
Bristol-Myers Squibb |
| ddI, didanosine |
Videx EC (enteric-coated) |
Bristol-Myers Squibb |
| FTC, emtricitabine |
FTC is only available in Canada co-formulated with tenofovir, as Truvada |
Gilead Sciences |
| tenofovir*
|
Viread |
Gilead Sciences |
| 3TC, lamivudine |
3TC |
ViiV Healthcare (formerly GlaxoSmithKline-Shire BioChem) |
| Non-Nukes (NNRTIs) |
| Common Name |
Brand Name |
Manufacturer |
| delavirdine |
Rescriptor |
ViiV Healthcare (formerly Pfizer) |
| efavirenz |
Sustiva |
Bristol-Myers Squibb |
| etravirine |
Intelence |
Tibotec |
| nevirapine |
Viramune |
Boehringer Ingelheim |
| Integrase Inhibitor |
| Common Name |
Brand Name |
Manufacturer |
| raltegravir |
Isentress |
Merck |
| Protease Inhibitors |
| Common Name |
Brand Name |
Manufacturer |
| atazanavir |
Reyataz |
Bristol-Myers Squibb |
| darunavir |
Prezista |
Tibotec |
| fosamprenavir |
Telzir |
ViiV Healthcare (formerly GlaxoSmithKline) |
| indinavir |
Crixivan |
Merck |
| lopinavir-ritonavir |
Kaletra |
Abbott Laboratories |
| nelfinavir |
Viracept |
ViiV Healthcare (formerly Pfizer) |
| ritonavir |
Norvir |
Abbott Laboratories |
| saquinavir |
Invirase |
Hoffmann-La Roche |
| tipranavir |
Aptivus |
Boehringer Ingelheim |
|
Co-Formulations Co-formulations take two or more different drugs and combine them into a single pill, reducing the number of pills that need to be taken.
|
| Common Name |
Brand Name |
Manufacturer |
| Atripla |
efavirenz + FTC + tenofovir |
Bristol Myers-Squibb/Gilead Sciences |
| Combivir |
AZT + 3TC |
ViiV Healthcare (formerly GlaxoSmithKline) |
| Kaletra |
lopinavir + ritonavir |
Abbott Laboratories |
| Kivexa |
3TC + abacavir |
ViiV Healthcare (formerly GlaxoSmithKline) |
| Trizivir |
AZT + 3TC + abacavir |
ViiV Healthcare (formerly GlaxoSmithKline) |
| Truvada |
FTC + tenofovir |
Gilead Sciences |
|
* Strictly speaking, tenofovir (Viread) is not a nucleoside analogue but a very similar molecule called a nucleotide analogue. This is largely a fine technical distinction; in practice, most HIV-positive people and their doctors refer to tenofovir as a nucleoside. |
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